Structure activity Relationship

Human Glutamate Pyruvate Transaminase (GPT): Localization to 8q24.3, cDNA and Genomic Sequences, and Polymorphic Sites

Information Systems / Genetics / Genomics / Polymorphism / Humans / Animals / Epidermolysis Bullosa / Polymerase Chain Reaction / DNA sequence design / Genetic Map / Biological evolution / Genes / Protein Sequence Analysis / Rats / Fluorescent in situ hybridization / Isoenzymes / Physical Map / Genetic variation / Amino Acid Profile / Genome sequence / Amino Acid Sequence / Base Sequence / Structure activity Relationship / DNA marker / Alanine Transaminase / Animals / Epidermolysis Bullosa / Polymerase Chain Reaction / DNA sequence design / Genetic Map / Biological evolution / Genes / Protein Sequence Analysis / Rats / Fluorescent in situ hybridization / Isoenzymes / Physical Map / Genetic variation / Amino Acid Profile / Genome sequence / Amino Acid Sequence / Base Sequence / Structure activity Relationship / DNA marker / Alanine Transaminase

Chemometric Studies on Potential Larvicidal Compounds Against Aedes Aegypti

Medicinal Chemistry / Principal Component Analysis / Insecticides / Animals / Mosquito Control / Larva / Structure activity Relationship / Aedes / Molecular Structure / Larva / Structure activity Relationship / Aedes / Molecular Structure

De Novo Cyclic Pseudopeptides Containing Aza-β 3 -amino Acids Exhibiting Antimicrobial Activities

Organic Chemistry / Medicinal Chemistry / Peptidomimetics / Sheep / Animals / Cyclic peptides / Gram Positive Bacteria / Amino Acids / Gram-negative bacteria / Anti-Bacterial Agents / Microbial Sensitivity Tests / Structure activity Relationship / Hemolysis / Cyclic peptides / Gram Positive Bacteria / Amino Acids / Gram-negative bacteria / Anti-Bacterial Agents / Microbial Sensitivity Tests / Structure activity Relationship / Hemolysis

In vitro activities of the multifunctional RNA silencing polymerase QDE-1 of Neurospora crassa

Biological Chemistry / RNA silencing / Neurospora crassa / Biological Sciences / CHEMICAL SCIENCES / Substrate Specificity / Structure activity Relationship / Substrate Specificity / Structure activity Relationship

Low molecular mass peptide dendrimers that express antimicrobial properties

Organic Chemistry / Escherichia coli / Staphylococcus aureus / Peptides / High Pressure Liquid Chromatography / Liquid Chromatography / Electrospray Ionization Mass Spectrometry / Anti-Bacterial Agents / Microbial Sensitivity Tests / Structure activity Relationship / Liquid Chromatography / Electrospray Ionization Mass Spectrometry / Anti-Bacterial Agents / Microbial Sensitivity Tests / Structure activity Relationship

Amino acid residue 247 in canine sulphotransferase SULT1D1: a new determinant of substrate selectivity

Biological Sciences / Dopamine / Dogs / Mutation / Animals / Biochemical / D-Aspartic Acid / CHEMICAL SCIENCES / Amino Acids / Substrate Specificity / Amino Acid Profile / Structure activity Relationship / Recombinant Proteins / Biochemical / D-Aspartic Acid / CHEMICAL SCIENCES / Amino Acids / Substrate Specificity / Amino Acid Profile / Structure activity Relationship / Recombinant Proteins

Scanning Alanine Mutagenesis and De-peptidization of a Candida albicans Myristoyl-CoA:Protein N-Myristoyltransferase Octapeptide Substrate Reveals Three Elements Critical for Molecular Recognition

Kinetics / Biological Chemistry / Biological Sciences / Candida albicans / CHEMICAL SCIENCES / Substrate Specificity / Alanine / Amino Acid Sequence / Structure activity Relationship / Recombinant Proteins / Substrate Specificity / Alanine / Amino Acid Sequence / Structure activity Relationship / Recombinant Proteins

Antimalarial Pyrido[1,2- a ]benzimidazoles

Organic Chemistry / Medicinal Chemistry / Malaria / Humans / Mice / Animals / Male / Rats / Plasmodium falciparum / Antimalarials / Pyridines / Benzimidazoles / Structure activity Relationship / Plasmodium berghei / Animals / Male / Rats / Plasmodium falciparum / Antimalarials / Pyridines / Benzimidazoles / Structure activity Relationship / Plasmodium berghei

3,4-Dihydropyrimido(1,2-a)indol-10(2H)-ones as potent non-peptidic inhibitors of caspase-3

Organic Chemistry / Apoptosis / Cell line / Stroke / Escherichia coli / Signal Transduction Pathway Models / Caspase / Protease Inhibitors / Bioorganic and medicinal Chemistry / Structure activity Relationship / Signal Transduction Pathway Models / Caspase / Protease Inhibitors / Bioorganic and medicinal Chemistry / Structure activity Relationship

Dipeptidyl peptidase IV-like molecules: homologous proteins or homologous activities?

Cell Migration / Membrane Proteins / Signal Transduction / Biological Sciences / Humans / Protein Turnover / Animals / Physical sciences / Enzyme / T lymphocytes / Human immunodeficiency virus / Isoenzymes / Enzyme activity / Structure activity Relationship / Dimerization / Protein Turnover / Animals / Physical sciences / Enzyme / T lymphocytes / Human immunodeficiency virus / Isoenzymes / Enzyme activity / Structure activity Relationship / Dimerization

Novel sulfonylurea derivatives as H3 receptor antagonists. Preliminary SAR studies

Organic Chemistry / Humans / Structure activity Relationship

Vanadium polypyridyl compounds as potential antiparasitic and antitumoral agents: New achievements

Inorganic Chemistry / Leishmania / Inorganic / Apoptosis / DNA / Humans / Chagas disease / Vanadium / Trypanosoma Cruzi / Trypanocidal Agents / Inorganic Biochemistry / Structure activity Relationship / Cell Survival / Antineoplastic Agents / Humans / Chagas disease / Vanadium / Trypanosoma Cruzi / Trypanocidal Agents / Inorganic Biochemistry / Structure activity Relationship / Cell Survival / Antineoplastic Agents

Physico-chemical characterization of a novel group of dopamine D3/D2 receptor ligands, potential atypical antipsychotic agents

Analytical Chemistry / Water / Linear models / Multivariate Analysis / Dopamine / Vitamin D receptor / Blood brain barrier / Animals / Partition Coefficient / High Pressure Liquid Chromatography / Analytical Method / Rats / Surface Area / Time Factors / Structural Properties / Atypical Antipsychotics / Reproducibility of Results / Wistar Rats / Linear Regression / Structure activity Relationship / Physico chemical Properties / Ligands / Molecular Structure / Piperidines / Vitamin D receptor / Blood brain barrier / Animals / Partition Coefficient / High Pressure Liquid Chromatography / Analytical Method / Rats / Surface Area / Time Factors / Structural Properties / Atypical Antipsychotics / Reproducibility of Results / Wistar Rats / Linear Regression / Structure activity Relationship / Physico chemical Properties / Ligands / Molecular Structure / Piperidines

3-Oxa-15-cyclohexyl prostaglandin DP receptor agonists as topical antiglaucoma agents

Organic Chemistry / Phase I clinical trial design / Glaucoma / Animals / Intraocular Pressure / Topical Drug Administration / Bioorganic and medicinal Chemistry / Rabbits / Hydrogen Atom / Structure activity Relationship / Protein Binding / Prostaglandin E2 / Molecular Structure / Topical Drug Administration / Bioorganic and medicinal Chemistry / Rabbits / Hydrogen Atom / Structure activity Relationship / Protein Binding / Prostaglandin E2 / Molecular Structure

On peroxide antimalarials

Multidrug Resistance / Natural Product / CHEMICAL SCIENCES / Plasmodium falciparum / Structure activity Relationship

5-Benzylidene 1,2-Dihydrochromeno[3,4- f ]quinolines, A Novel Class of Nonsteroidal Human Progesterone Receptor Agonists

Organic Chemistry / Medicinal Chemistry / Macromolecular X-Ray Crystallography / Progesterone / Humans / Female / Animals / Rats / Medicinal / Quinolines / Structure activity Relationship / Uterus / Ovariectomy / Female / Animals / Rats / Medicinal / Quinolines / Structure activity Relationship / Uterus / Ovariectomy

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