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Structure activity Relationship
Structure activity Relationship
Effects of selected pharmaceutical products on phagocytic activity in Elliptio complanata mussels
Cell Adhesion / Crop Physiology and Biochemistry / Biological Sciences / Environmental Sciences / Bivalvia / Nitric oxide / Animals / Lipid peroxidation / Hemocytes / Immune system / Phagocytosis / Carbamazepine / Freshwater pearl mussel / Functional Group / Esterases / Domestic Wastewater / Structure activity Relationship / Nitric oxide / Animals / Lipid peroxidation / Hemocytes / Immune system / Phagocytosis / Carbamazepine / Freshwater pearl mussel / Functional Group / Esterases / Domestic Wastewater / Structure activity Relationship
2-(Arylpropionylamino)- and 2-(arylacryloylamino)benzophenones: farnesyltransferase inhibition and antimalarial activity
Mass Spectrometry / Magnetic Resonance Spectroscopy / Humans / Escherichia coli / Animals / Pharmazie / Benzophenones / Plasmodium falciparum / Antimalarials / Thiazoles / Structure activity Relationship / Pharmazie / Benzophenones / Plasmodium falciparum / Antimalarials / Thiazoles / Structure activity Relationship
Light curable dental composites designed with colloidal crystal reinforcement
Engineering / Crystallization / Dental Materials / Elasticity / Compressive Strength / Colloids / Hardness / Composite resins / Dental Stress Analysis / Polymethyl Methacrylates / Materials Testing / Structure activity Relationship / Silicon Dioxide / Polyethylene Glycols / Colloids / Hardness / Composite resins / Dental Stress Analysis / Polymethyl Methacrylates / Materials Testing / Structure activity Relationship / Silicon Dioxide / Polyethylene Glycols
Female sex pheromone of Cameraria ohridella Desch. and Dim. (Lepidoptera: Gracillariidae): structure confirmation, synthesis and biological activity of (8E,10Z)-8,10-tetradecadienal and some analogues
Female / Animals / Gas Chromatography / Moths / Structure activity Relationship / Molecular Structure / Plant Leaves / Molecular Structure / Plant Leaves
Amphibian antimicrobial peptides and Protozoa: Lessons from parasites
Chemical Engineering / Phospholipids / Biological Sciences / Animals / Physical sciences / Antimicrobial Peptide / Antimicrobial Cationic Peptides / Amino Acid Sequence / Body of Knowledge / Structure activity Relationship / Plasma Membrane / Biochemistry and cell biology / Amphibian Proteins / Antimicrobial Peptide / Antimicrobial Cationic Peptides / Amino Acid Sequence / Body of Knowledge / Structure activity Relationship / Plasma Membrane / Biochemistry and cell biology / Amphibian Proteins
Identification of key amino acid residues in Neisseria polysaccharea amylosucrase
Catalysis / Glycoside hydrolase / Protein Structure and Function / Sequence alignment / Glutathione / Neisseria / D-Aspartic Acid / Enzyme / Amino Acids / Amino Acid Profile / Amino Acid Sequence / Base Sequence / Structure activity Relationship / Polyacrylamide Gel Electrophoresis / Enzymatic Activity / Site-directed Mutagenesis / Glutamic Acid / Histidine / Biochemistry and cell biology / Neisseria / D-Aspartic Acid / Enzyme / Amino Acids / Amino Acid Profile / Amino Acid Sequence / Base Sequence / Structure activity Relationship / Polyacrylamide Gel Electrophoresis / Enzymatic Activity / Site-directed Mutagenesis / Glutamic Acid / Histidine / Biochemistry and cell biology
Microbicidal effect of the lactoferrin peptides Lactoferricin17–30, Lactoferrampin265–284, and Lactoferrin chimera on the parasite Entamoeba histolytica
Growth Kinetics / Ulcerative colitis / Animals / Parasites / Peptides / Anti-Bacterial Agents / Biometals / Entamoeba histolytica / Amino Acid Profile / Structure activity Relationship / Biochemistry and cell biology / Anti-Bacterial Agents / Biometals / Entamoeba histolytica / Amino Acid Profile / Structure activity Relationship / Biochemistry and cell biology
Comparison of anorexigenic and behavioral potency of phenylethylamines
Animal Behavior / Animals / Methamphetamine / Male / Experimental Pharmacology / Amphetamine / Food habits / Rats / Chlorine / Structure activity Relationship / Fenfluramine / Phentermine / Amphetamine / Food habits / Rats / Chlorine / Structure activity Relationship / Fenfluramine / Phentermine
Engineering a terbium-binding site into an integral membrane protein for luminescence energy transfer
Fluorescence / Multidisciplinary / Protein Engineering / Fluorescence Resonance Energy Transfer / Mutation / Escherichia coli / Terbium / Membrane transport proteins / Protein Secondary Structure Prediction / Spectrum analysis / Energy Transfer / Membrane Protein / Structure activity Relationship / Cytoplasm / Binding Site / Escherichia coli / Terbium / Membrane transport proteins / Protein Secondary Structure Prediction / Spectrum analysis / Energy Transfer / Membrane Protein / Structure activity Relationship / Cytoplasm / Binding Site
Parthenolide Inhibits Tubulin Carboxypeptidase Activity
Principal Component Analysis / Cancer / Drug interactions / Cell Division / Humans / NF-kappa B / Paclitaxel / Sesquiterpenes / HeLa cells / Tubulin / Carboxypeptidases / Structure activity Relationship / Tumor Progression / NF-kappa B / Paclitaxel / Sesquiterpenes / HeLa cells / Tubulin / Carboxypeptidases / Structure activity Relationship / Tumor Progression
Partial repair of deamidation-damaged calmodulin by protein carboxyl methyltransferase
Membranes / Biological Chemistry / DNA repair / Biological Sciences / Brain / Methylation / Animals / High Pressure Liquid Chromatography / CHEMICAL SCIENCES / Cattle / Calmodulin / Structure activity Relationship / Hydrogen-Ion Concentration / Methylation / Animals / High Pressure Liquid Chromatography / CHEMICAL SCIENCES / Cattle / Calmodulin / Structure activity Relationship / Hydrogen-Ion Concentration
Antiviral evaluation of N-amino-1,2,3-triazoles against Cantagalo virus replication in cell culture
Organic Chemistry / Cell Culture / Cercopithecus aethiops / Cell line / Animals / European / Vaccinia Virus / Microbial Sensitivity Tests / Structure activity Relationship / X Ray Crystallography / Cell Survival / Antiviral Agents / Molecular Structure / European / Vaccinia Virus / Microbial Sensitivity Tests / Structure activity Relationship / X Ray Crystallography / Cell Survival / Antiviral Agents / Molecular Structure
X-L INKED L YMPHOPROLIFERATIVE D ISEASE : A Progressive Immunodeficiency
Immunology / Transcription Factors / Signal Transduction / Humans / Sequence alignment / Male / Phenotype / Respiratory Tract Infections / Diffuse Large B-Cell Lymphoma / Disease Progression / Protein Conformation / Amino Acid Sequence / Structure activity Relationship / Antigen presenting cells / Agammaglobulinemia / Male / Phenotype / Respiratory Tract Infections / Diffuse Large B-Cell Lymphoma / Disease Progression / Protein Conformation / Amino Acid Sequence / Structure activity Relationship / Antigen presenting cells / Agammaglobulinemia
Identification of 2-hydroxymethyl-4-[5-(4-methoxyphenyl)-3-trifluoromethyl-pyrazol-1-yl]-N-propionylbenzenesulfonamide sodium as a potential COX-2 inhibitor for oral and parenteral administration
Organic Chemistry / Enzyme Inhibitors / Prodrugs / Humans / Animals / Male / Solubility / Rats / Edema / Fever / Foot / Wistar Rats / Carrageenan / Water soluble polymers / Bioorganic and medicinal Chemistry / Structure activity Relationship / Hyperalgesia / Endotoxins / Molecular Structure / Male / Solubility / Rats / Edema / Fever / Foot / Wistar Rats / Carrageenan / Water soluble polymers / Bioorganic and medicinal Chemistry / Structure activity Relationship / Hyperalgesia / Endotoxins / Molecular Structure
An Aberrant Sequence in a Connexin46 Mutant Underlies Congenital Cataracts
Gap Junctions / Flow Cytometry / Biological Chemistry / Gene expression / Biological Sciences / Xenopus / Humans / Mutation / Mice / Animals / Biological / Cataract / CHEMICAL SCIENCES / Fluorescent Antibody Technique / HeLa cells / Transfection / Amino Acid Sequence / Oocytes / Structure activity Relationship / Electric Conductivity / Xenopus / Humans / Mutation / Mice / Animals / Biological / Cataract / CHEMICAL SCIENCES / Fluorescent Antibody Technique / HeLa cells / Transfection / Amino Acid Sequence / Oocytes / Structure activity Relationship / Electric Conductivity
Xanthones as Potential Antioxidants
Antioxidants / Humans / Structure activity Relationship / Oxidation-Reduction
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