Enzyme Inhibitors

Identification of 2-hydroxymethyl-4-[5-(4-methoxyphenyl)-3-trifluoromethyl-pyrazol-1-yl]-N-propionylbenzenesulfonamide sodium as a potential COX-2 inhibitor for oral and parenteral administration

Organic Chemistry / Enzyme Inhibitors / Prodrugs / Humans / Animals / Male / Solubility / Rats / Edema / Fever / Foot / Wistar Rats / Carrageenan / Water soluble polymers / Bioorganic and medicinal Chemistry / Structure activity Relationship / Hyperalgesia / Endotoxins / Molecular Structure / Male / Solubility / Rats / Edema / Fever / Foot / Wistar Rats / Carrageenan / Water soluble polymers / Bioorganic and medicinal Chemistry / Structure activity Relationship / Hyperalgesia / Endotoxins / Molecular Structure

Cefcapene inactivates chromosome-encoded class C β-lactamases

Kinetics / Enzyme Inhibitors / Escherichia coli / Cephalosporins / Pseudomonas aeruginosa / Enzyme / Steady state / Pseudomonas Aeruginosa / Drug Stability / Kinetic Parameter / Beta Lactamases / Enzyme / Steady state / Pseudomonas Aeruginosa / Drug Stability / Kinetic Parameter / Beta Lactamases

Antiviral prophylaxis during pandemic influenza may increase drug resistance

Microbiology / Medical Microbiology / Enzyme Inhibitors / Disease Outbreaks / Uncertainty / Humans / Computer Simulation / Pandemic Influenza / Drug Resistance / Social distance / Neuraminidase / Clinical Sciences / Prevalence / Basic Reproduction Number / Antiviral Agents / Humans / Computer Simulation / Pandemic Influenza / Drug Resistance / Social distance / Neuraminidase / Clinical Sciences / Prevalence / Basic Reproduction Number / Antiviral Agents

Novel Hydroxysteroid (17β) Dehydrogenase 1 Inhibitors Reverse Estrogen-Induced Endometrial Hyperplasia in Transgenic Mice

Enzyme Inhibitors / Transgenic Mice / Humans / Mice / Female / Animals / Estrogens / Uterus / Progestins / Estradiol / Endometrial Hyperplasia / Animals / Estrogens / Uterus / Progestins / Estradiol / Endometrial Hyperplasia

Unsuccessful intraventricular pentosan polysulphate treatment of variant Creutzfeldt-Jakob disease

Magnetic Resonance Imaging / Enzyme Inhibitors / Biopsy / Brain / Humans / Female / Mental Disorders / Clinical Sciences / Prions / Adult / Disease Progression / Seizures / Neurosciences / Cognition disorders / Female / Mental Disorders / Clinical Sciences / Prions / Adult / Disease Progression / Seizures / Neurosciences / Cognition disorders

Amino hydroxamic acids as potent inhibitors of leukotriene A4 hydrolase

Organic Chemistry / Enzyme Inhibitors / Magnetic Resonance Spectroscopy / Humans / Zinc / Enzyme / Bioorganic and medicinal Chemistry / Chelating Agents / Hydroxamic Acids / Enzyme / Bioorganic and medicinal Chemistry / Chelating Agents / Hydroxamic Acids

Differential expression of α1-adrenergic receptor subtypes in coronary microvascular endothelial cells in culture

Enzyme Inhibitors / Endothelial Cells / Nitric oxide / Animals / Male / European / Rats / Nitric Oxide Synthase / Endothelial cell / Wistar Rats / Phenylephrine / Blood Vessel / Intracellular Calcium / Immunoblotting / Bradykinin / European / Rats / Nitric Oxide Synthase / Endothelial cell / Wistar Rats / Phenylephrine / Blood Vessel / Intracellular Calcium / Immunoblotting / Bradykinin

Mifepristone attenuates human chorionic gonadotropin–induced extracellular signal–regulated kinase 1/2 phosphorylation, cyclooxygenase-2, and prostaglandin E2 production in human granulosa luteal cells

Drug interactions / Enzyme Inhibitors / Flavonoids / Humans / Fertility and Sterility / Female / Phosphorylation / Mitogen Activated Protein Kinase / Clinical Sciences / Adult / Public health systems and services research / Down-Regulation / Female / Phosphorylation / Mitogen Activated Protein Kinase / Clinical Sciences / Adult / Public health systems and services research / Down-Regulation

Physiological and genetic responses of European eel (Anguilla anguilla L.) to short-term chromium or copper exposure?Influence of preexposure to a PAH-like compound

Genetics / Environmental Toxicology / Enzyme Inhibitors / DNA damage / Biological Sciences / Environmental Sciences / Blood Glucose / Copper / Animals / Thyroid Hormones / Chromium / European eel / CHEMICAL SCIENCES / Anguilla anguilla / The Endocrine System Function / Anguilla / Environmental Exposure / Environmental Sciences / Blood Glucose / Copper / Animals / Thyroid Hormones / Chromium / European eel / CHEMICAL SCIENCES / Anguilla anguilla / The Endocrine System Function / Anguilla / Environmental Exposure

Physiological and genetic responses of European eel (Anguilla anguilla L.) to short-term chromium or copper exposure?Influence of preexposure to a PAH-like compound

Genetics / Environmental Toxicology / Enzyme Inhibitors / DNA damage / Biological Sciences / Environmental Sciences / Blood Glucose / Copper / Animals / Thyroid Hormones / Chromium / European eel / CHEMICAL SCIENCES / Anguilla anguilla / The Endocrine System Function / Anguilla / Environmental Exposure / Environmental Sciences / Blood Glucose / Copper / Animals / Thyroid Hormones / Chromium / European eel / CHEMICAL SCIENCES / Anguilla anguilla / The Endocrine System Function / Anguilla / Environmental Exposure

Hypoxia sustains glioblastoma radioresistance through ERKs/DNA-PKcs/HIF-1α functional interplay

Oncology / Enzyme Inhibitors / Humans / Nitriles / Glioblastoma / Oxygen / Radiation Tolerance / Benzamides / Oxygen / Radiation Tolerance / Benzamides

Aminoacyl-tRNA synthetase inhibitors as potential antibiotics

Organic Chemistry / Medicinal Chemistry / Drug Discovery / Enzyme Inhibitors / Humans / Animals / Anti-Bacterial Agents / Animals / Anti-Bacterial Agents

Intrarenal Aminopeptidase N Inhibition Augments Natriuretic Responses to Angiotensin III in Angiotensin Type 1 Receptor-Blocked Rats

Enzyme Inhibitors / Hypertension / Animals / Behavioral Animal Models / Clinical Sciences / Rats / Sodium / Methionine / Benzimidazoles / Angiotensin II / Cumulant / Rats / Sodium / Methionine / Benzimidazoles / Angiotensin II / Cumulant

Intrarenal Aminopeptidase N Inhibition Augments Natriuretic Responses to Angiotensin III in Angiotensin Type 1 Receptor-Blocked Rats

Enzyme Inhibitors / Hypertension / Animals / Behavioral Animal Models / Clinical Sciences / Rats / Sodium / Methionine / Benzimidazoles / Angiotensin II / Cumulant / Rats / Sodium / Methionine / Benzimidazoles / Angiotensin II / Cumulant

Acetylcholinesterases from Elapidae snake venoms: biochemical, immunological and enzymatic characterization

Catalysis / Enzyme Inhibitors / Biological Sciences / Physical sciences / Acetylcholinesterase / Monoclonal Antibodies / Affinity chromatography / Enzyme / Snake Venom / Active site / Protein Conformation / Monoclonal Antibody / Bovine Serum Albumin / Monoclonal Antibodies / Affinity chromatography / Enzyme / Snake Venom / Active site / Protein Conformation / Monoclonal Antibody / Bovine Serum Albumin

Protein Kinase A Activation Promotes Plasma Membrane Insertion of DCC from an Intracellular Pool: A Novel Mechanism Regulating Commissural Axon Extension

Neuroscience / Enzyme Inhibitors / Molecular Mechanics / cyclic AMP / Animals / Spinal Cord / P-glycoprotein / Axon Guidance / The / Rats / Exocytosis / Axons / Plasma Membrane / Protein Transport / Cell Adhesion Molecules / Axon Outgrowth / Spinal Cord / P-glycoprotein / Axon Guidance / The / Rats / Exocytosis / Axons / Plasma Membrane / Protein Transport / Cell Adhesion Molecules / Axon Outgrowth

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