In Vitro

Efficacy of Ciprofloxacin and Moxifloxacin against Nocardia brasiliensis In Vitro and in an Experimental Model of Actinomycetoma in BALB/c Mice

Pharmacology / Microbiology / Pharmacy / Medical Microbiology / In Vitro / Models / Mice / Female / Animals / Bacteria / Antimicrobial agents / Microbial Sensitivity Tests / Mycetoma / Ciprofloxacin / Quinolines / Nocardia / Fluoroquinolones / Experimental Model / Models / Mice / Female / Animals / Bacteria / Antimicrobial agents / Microbial Sensitivity Tests / Mycetoma / Ciprofloxacin / Quinolines / Nocardia / Fluoroquinolones / Experimental Model

Enhancement of pharmacokinetic properties and in vivo efficacy of benzylidene ketal M2 muscarinic receptor antagonists via benzamide modification

Organic Chemistry / Pharmacokinetics / In Vitro / Humans / Animals / Drug Design / Acetylcholine / Bioavailability / Microdialysis / In Vivo / Rats / Rat / Cholinergic Receptor / Bioorganic and medicinal Chemistry / Structure activity Relationship / Muscarinic Receptor / Chemical Synthesis / Area Under Curve / Benzamides / Drug Design / Acetylcholine / Bioavailability / Microdialysis / In Vivo / Rats / Rat / Cholinergic Receptor / Bioorganic and medicinal Chemistry / Structure activity Relationship / Muscarinic Receptor / Chemical Synthesis / Area Under Curve / Benzamides

Antimalarial Agents from Plants. III. Trichothecenes from Ficus fistulosa and Rhaphidophora decursiva

Complementary and Alternative Medicine / Plant Biology / Pharmacognosy / In Vitro / Animals / STEM / Araceae / Ficus / Bark / Isolation / Plant extracts / Plasmodium falciparum / Antimalarials / Biological activity / Extract / Active Ingredient / Planta / Molecular Structure / Plant Leaves / Terpenoid / STEM / Araceae / Ficus / Bark / Isolation / Plant extracts / Plasmodium falciparum / Antimalarials / Biological activity / Extract / Active Ingredient / Planta / Molecular Structure / Plant Leaves / Terpenoid

New vasorelaxant indole alkaloids, villocarines A–D from Uncaria villosa

Organic Chemistry / Calcium / Pharmacognosy / Magnetic Resonance Spectroscopy / Structural Analysis / In Vitro / Endothelial Cells / Nitric oxide / Animals / Calcium channels / Potassium / Isolation / Rats / Endothelial cell / Rat / Voltage-Gated Potassium Channels / Molecular Conformation / Bioorganic and medicinal Chemistry / Biological activity / Uncaria / Aorta / Indole Alkaloids / Plant Leaves / In Vitro / Endothelial Cells / Nitric oxide / Animals / Calcium channels / Potassium / Isolation / Rats / Endothelial cell / Rat / Voltage-Gated Potassium Channels / Molecular Conformation / Bioorganic and medicinal Chemistry / Biological activity / Uncaria / Aorta / Indole Alkaloids / Plant Leaves

Contamination and effects of perfluorochemicals in baikal seal (Pusa sibirica). 1. Residue level, tissue distribution, and temporal trend

Multidisciplinary / Environmental science and technology / In Vitro / Liver / Animals / Peroxisome proliferator-activated receptor / Molecular Characterization / Real Time system / Base Sequence / Sensitivity and Specificity / Environmental / Peroxisome proliferator-activated receptor / Molecular Characterization / Real Time system / Base Sequence / Sensitivity and Specificity / Environmental

Antimalarial in-vivo activity of bis(9-amino-6-chloro-2-methoxyacridines)

Pharmacy / Malaria / In Vitro / Toxicity / Mice / Pharmacology and Clinical pharmacy / Female / Animals / Antimalarials / Alkylation / Acylation / Biological activity / Chloroquine / Chemical Synthesis / Plasmodium berghei / Pharmacology and Clinical pharmacy / Female / Animals / Antimalarials / Alkylation / Acylation / Biological activity / Chloroquine / Chemical Synthesis / Plasmodium berghei

Antimicrobial activity of Terminalia macroptera root

Complementary and Alternative Medicine / Plant Biology / Ethnopharmacology / Pharmacognosy / Medicinal Plants / In Vitro / ROOT / Infectious Disease / Escherichia coli / Vibrio cholerae / Antimicrobial activity / Bacteria / Ethanol / Candida albicans / Enterobacteriaceae / Plant Roots / Guinea Bissau / Anti-Bacterial Agents / Plant extracts / Microbial Sensitivity Tests / Biological activity / Extract / Medicinal Plant / Minimum inhibitory concentration / Thallophyta / In Vitro / ROOT / Infectious Disease / Escherichia coli / Vibrio cholerae / Antimicrobial activity / Bacteria / Ethanol / Candida albicans / Enterobacteriaceae / Plant Roots / Guinea Bissau / Anti-Bacterial Agents / Plant extracts / Microbial Sensitivity Tests / Biological activity / Extract / Medicinal Plant / Minimum inhibitory concentration / Thallophyta

Unusual antimalarial meroditerpenes from tropical red macroalgae

Organic Chemistry / Drug Discovery / Pharmacognosy / Structural Analysis / In Vitro / Humans / Circular Dichroism / Natural Product / Seaweed / Isolation / Absolute Configuration / Diterpenes / Plasmodium falciparum / Antimalarials / Conformational Analysis / Biological activity / Terpenoid / Humans / Circular Dichroism / Natural Product / Seaweed / Isolation / Absolute Configuration / Diterpenes / Plasmodium falciparum / Antimalarials / Conformational Analysis / Biological activity / Terpenoid

ChemInform Abstract: Unusual Antimalarial Meroditerpenes from Tropical Red Macroalgae

Organic Chemistry / Drug Discovery / Pharmacognosy / Structural Analysis / In Vitro / Humans / Circular Dichroism / Natural Product / Seaweed / Isolation / Absolute Configuration / Diterpenes / Plasmodium falciparum / Antimalarials / Conformational Analysis / Biological activity / Terpenoid / Humans / Circular Dichroism / Natural Product / Seaweed / Isolation / Absolute Configuration / Diterpenes / Plasmodium falciparum / Antimalarials / Conformational Analysis / Biological activity / Terpenoid

Unusual antimalarial meroditerpenes from tropical red macroalgae

Organic Chemistry / Drug Discovery / Pharmacognosy / Structural Analysis / In Vitro / Humans / Circular Dichroism / Natural Product / Seaweed / Isolation / Absolute Configuration / Diterpenes / Plasmodium falciparum / Antimalarials / Conformational Analysis / Biological activity / Terpenoid / Humans / Circular Dichroism / Natural Product / Seaweed / Isolation / Absolute Configuration / Diterpenes / Plasmodium falciparum / Antimalarials / Conformational Analysis / Biological activity / Terpenoid

Antibacterial activity of hydro-alcoholic extract leaves of jambolan (Syzygium cumini (L.) Skells)

In Vitro / Gram Positive / Antimicrobial activity / Antibacterial activity / Gram-negative bacteria / Leaves / Medicinal Plant / Multiple Drug Resistance / Leaves / Medicinal Plant / Multiple Drug Resistance

Bone sialoprotein deficiency impairs osteoclastogenesis and mineral resorption in vitro

Engineering / Minerals / Apoptosis / Biological Sciences / Spleen / In Vitro / Cell Differentiation / Humans / Mice / Bone / Animals / Osteoclasts / Osteopontin / Bone Mineral Density / Dentin / Biological markers / Osteogenesis / Cell Proliferation / BSP / Durapatite / Somatic Cell Count / Recombinant Proteins / Resorption / Bone Resorption / Gene expression profiling / In Vitro / Cell Differentiation / Humans / Mice / Bone / Animals / Osteoclasts / Osteopontin / Bone Mineral Density / Dentin / Biological markers / Osteogenesis / Cell Proliferation / BSP / Durapatite / Somatic Cell Count / Recombinant Proteins / Resorption / Bone Resorption / Gene expression profiling

A hybrid numerical method to compute erythrocyte TMP in low-frequency electric fields

Algorithms / Information Science / Biomedical Engineering / Finite Element Methods / Finite element method / Boundary Element Methods / Low Frequency / Numerical Method / Finite Element Analysis / In Vitro / Humans / Computer Simulation / Boundary Element Method / Electromagnetic Fields / Three Dimensional / Erythrocyte Membrane / Erythrocytes / Electric Field / Electrical And Electronic Engineering / Extracellular / Hybrid Method / Boundary Element Methods / Low Frequency / Numerical Method / Finite Element Analysis / In Vitro / Humans / Computer Simulation / Boundary Element Method / Electromagnetic Fields / Three Dimensional / Erythrocyte Membrane / Erythrocytes / Electric Field / Electrical And Electronic Engineering / Extracellular / Hybrid Method

Antimicrobial activity of Terminalia macroptera root

Complementary and Alternative Medicine / Plant Biology / Ethnopharmacology / Pharmacognosy / Medicinal Plants / In Vitro / ROOT / Infectious Disease / Escherichia coli / Vibrio cholerae / Antimicrobial activity / Bacteria / Ethanol / Candida albicans / Enterobacteriaceae / Plant Roots / Guinea Bissau / Anti-Bacterial Agents / Plant extracts / Microbial Sensitivity Tests / Biological activity / Extract / Medicinal Plant / Minimum inhibitory concentration / Thallophyta / In Vitro / ROOT / Infectious Disease / Escherichia coli / Vibrio cholerae / Antimicrobial activity / Bacteria / Ethanol / Candida albicans / Enterobacteriaceae / Plant Roots / Guinea Bissau / Anti-Bacterial Agents / Plant extracts / Microbial Sensitivity Tests / Biological activity / Extract / Medicinal Plant / Minimum inhibitory concentration / Thallophyta
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