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Organic Chemistry
Organic Chemistry
Simple and effective synthesis of pentamethylcyclopentadienyl oxo-peroxo and dioxo tungsten acetylide complexes
Inorganic Chemistry / Organic Chemistry / Organometallic Chemistry / Hydrogen Peroxide / X ray diffraction / Room Temperature / Single Crystal / Room Temperature / Single Crystal
In vitro and in vivo profile of 5-[(4′-trifluoromethyl-biphenyl-2-carbonyl)-amino]-1H-indole-2-carboxylic acid benzylmethyl carbamoylamide (dirlotapide), a novel potent MTP inhibitor for obesity
Organic Chemistry / Medicinal Chemistry / Obesity / Pharmaceutical Chemistry / Dogs / Humans / Animals / Drug Design / Enzyme / Food intake / Rats / Carboxylic Acids / Molecular Conformation / Bioorganic and medicinal Chemistry / Hydrogen-Ion Concentration / Carbamates / Humans / Animals / Drug Design / Enzyme / Food intake / Rats / Carboxylic Acids / Molecular Conformation / Bioorganic and medicinal Chemistry / Hydrogen-Ion Concentration / Carbamates
Chemistry of Petrochemical processes MATAR
Environmental Engineering / Chemical Engineering / Organic Chemistry
5-Benzylidene 1,2-Dihydrochromeno[3,4- f ]quinolines, A Novel Class of Nonsteroidal Human Progesterone Receptor Agonists
Organic Chemistry / Medicinal Chemistry / Macromolecular X-Ray Crystallography / Progesterone / Humans / Female / Animals / Rats / Medicinal / Quinolines / Structure activity Relationship / Uterus / Ovariectomy / Female / Animals / Rats / Medicinal / Quinolines / Structure activity Relationship / Uterus / Ovariectomy
5-Aryl-1,2-dihydrochromeno[3,4- f ]quinolines: A Novel Class of Nonsteroidal Human Progesterone Receptor Agonists
Organic Chemistry / Medicinal Chemistry / Magnetic Resonance Spectroscopy / Humans / Female / Animals / Rats / Medicinal / Quinolines / Structure activity Relationship / Uterus / Animals / Rats / Medicinal / Quinolines / Structure activity Relationship / Uterus
A synthon approach to spiro compounds
Organic Chemistry / Tetrahedron
The efficiency of proton transfer in Kirby’s enzyme model, a computational approach
Organic Chemistry / Proton Transfer / Ab Initio Calculation
Polyelectrolyte Complexes
Materials Engineering / Organic Chemistry / Polymer science / Retinoic Acid
Acyl sulfonamide anti-proliferatives. Part 2: Activity of heterocyclic sulfonamide derivatives
Organic Chemistry / Humans / Bioorganic and medicinal Chemistry / Cell Proliferation / Structure activity Relationship / Vascular Endothelial Growth Factor
SUPERNOVA REMNANT KES 17: AN EFFICIENT COSMIC RAY ACCELERATOR INSIDE A MOLECULAR CLOUD
Organic Chemistry
Bicyclic glutamic acid derivatives
Analytical Chemistry / Organic Chemistry / Macromolecular X-Ray Crystallography / Chirality / Circular Dichroism / Cyclization / Hydrolysis / Esters / Glutamic Acid / *Hot Temperature / Molecular Structure / Solvents / Cyclization / Hydrolysis / Esters / Glutamic Acid / *Hot Temperature / Molecular Structure / Solvents
Preparation and Pharmacological Characterization of trans -2-Amino-5(6)-fluoro-6(5)-hydroxy-1-phenyl-2,3-dihydro-1 H -indenes as D 2 -like Dopamine Receptor Agonists
Organic Chemistry / Medicinal Chemistry / cyclic AMP / Animals / dopamine receptor D4 / Rats / Swine / Radioligand Assay / Medicinal / Structure activity Relationship / cyclic GMP / Rats / Swine / Radioligand Assay / Medicinal / Structure activity Relationship / cyclic GMP
SN 2005cg: Explosion Physics and Circumstellar Interaction of a Normal Type Ia Supernova in a Low-Luminosity Host
Organic Chemistry / Astrophysical Plasma / High Redshift Universe
Essential oil composition and antimicrobial activity of Ballota nigra L. ssp foetida
Organic Chemistry / Plant Biology
Application of Structure-Based Drug Design and Parallel Chemistry to Identify Selective, Brain Penetrant, In Vivo Active Phosphodiesterase 9A Inhibitors
Organic Chemistry / Medicinal Chemistry / Macromolecular X-Ray Crystallography / Dogs / Humans / Blood brain barrier / Animals / Drug Design / Rats / Pyrazoles / Structure activity Relationship / cyclic GMP / Molecular Structure / Blood brain barrier / Animals / Drug Design / Rats / Pyrazoles / Structure activity Relationship / cyclic GMP / Molecular Structure
New 7,8-ethylenedioxy-2,3-benzodiazepines as noncompetitive AMPA receptor antagonists
Organic Chemistry / Pharmaceutical Chemistry / Humans / Mice / DBA / Animals / Drug Design / Benzodiazepines / Rats / Bioorganic and medicinal Chemistry / Structure activity Relationship / Protein Binding / Functional Testing / Animals / Drug Design / Benzodiazepines / Rats / Bioorganic and medicinal Chemistry / Structure activity Relationship / Protein Binding / Functional Testing
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