Organic Chemistry

Fancy Bioisosteres:  Novel Paracyclophane Derivatives As Super-Affinity Dopamine D3 Receptor Antagonists

Organic Chemistry / Medicinal Chemistry / Magnetic Resonance Spectroscopy / Dopamine / Humans / Mutation / Animals / Amides / Swine / Radioligand Assay / Medicinal / Molecular Conformation / Structure activity Relationship / Mutation / Animals / Amides / Swine / Radioligand Assay / Medicinal / Molecular Conformation / Structure activity Relationship

Steroidal Indoxyls, Indoles, and Quinolines 1

Inorganic Chemistry / Organic Chemistry

CoMSIA and POM analyses of anti-malarial activity of synthetic prodiginines

Organic Chemistry / Quantitative Structure Activity Relationship / Prodigiosin / Antimalarials / Molecular Structure

Aza-bicyclic amino acid carboxamides as α4β1/α4β7 integrin receptor antagonists

Organic Chemistry / Multiple sclerosis / Rheumatoid Arthritis / Inflammatory Bowel Disease / Amino Acid Profile / Bioorganic and medicinal Chemistry

Aza-bicyclic amino acid sulfonamides as α4β1/α4β7 integrin antagonists

Organic Chemistry / Amino Acid Profile / Conformational Analysis / Biological activity

RGD Mimetics containing a central hydantoin scaffold: αVβ3 vs αIIbβ3 selectivity requirements

Organic Chemistry / Fibrinogen / Humans / Peptides / Bioorganic and medicinal Chemistry / Imidazoles / Protein Binding / Molecular Structure / Imidazoles / Protein Binding / Molecular Structure
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