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In vitro and in vivo comparison of two non-peptide tachykinin NK3 receptor antagonists: Improvements in efficacy achieved through enhanced brain penetration or altered pharmacological characteristics
Animal Behavior / Prefrontal Cortex / Nucleus Accumbens / Dopamine / Brain / Humans / Cerebral Cortex / Animals / Male / Central Nervous System / Peptides / Habenula / Neurons / Haloperidol / European / Microdialysis / Molecular cloning / Rats / Neuronal Activity / Guinea Pig / Substance P / Quinolines / Extracellular Space / Medial Prefrontal Cortex / Clinical evaluation / Humans / Cerebral Cortex / Animals / Male / Central Nervous System / Peptides / Habenula / Neurons / Haloperidol / European / Microdialysis / Molecular cloning / Rats / Neuronal Activity / Guinea Pig / Substance P / Quinolines / Extracellular Space / Medial Prefrontal Cortex / Clinical evaluation
In vitro and in vivo comparison of two non-peptide tachykinin NK3 receptor antagonists: Improvements in efficacy achieved through enhanced brain penetration or altered pharmacological characteristics
Animal Behavior / Neurotransmission / Pharmacokinetics / Comparative Study / Prefrontal Cortex / Nucleus Accumbens / Dopamine / In Vitro / Brain / Humans / Cerebral Cortex / Animals / Male / Central Nervous System / Peptides / Habenula / Neurons / Efficiency / Haloperidol / European / Microdialysis / Molecular cloning / In Vivo / Rats / Neuronal Activity / Guinea Pig / Substance P / Quinolines / Extracellular Space / Pharmacokinetic / Medial Prefrontal Cortex / Clinical evaluation / Inositol Phosphates / Nucleus Accumbens / Dopamine / In Vitro / Brain / Humans / Cerebral Cortex / Animals / Male / Central Nervous System / Peptides / Habenula / Neurons / Efficiency / Haloperidol / European / Microdialysis / Molecular cloning / In Vivo / Rats / Neuronal Activity / Guinea Pig / Substance P / Quinolines / Extracellular Space / Pharmacokinetic / Medial Prefrontal Cortex / Clinical evaluation / Inositol Phosphates
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