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Trypanocidal Agents
Trypanocidal Agents
Trypanocidal and Leishmanicidal Activities of Sesquiterpene Lactones from Ambrosia tenuifolia Sprengel (Asteraceae)
Microbiology / Medical Microbiology / Argentina / Medicinal Plants / Flavonoids / Lipopolysaccharide / Phytotherapy / Experimental parasitology / Humans / Infrared spectroscopy / Mice / Female / Animals / Natural Product / Male / Penaeus Monodon / Horseshoe crabs / Litopenaeus Vannamei / Peptides / Cyclic peptides / Selection Index / Antimicrobial Peptide / Chagas disease / Sesquiterpenes / T lymphocytes / Experimental / Infrared / Antimicrobial Cationic Peptides / Trypanosoma Cruzi / Cytotoxic Activity / Tritium / Eupatorium / Xenopus laevis / Antimicrobial agents / Mytilus edulis / Cutaneous Leishmaniasis / Veterinary Sciences / Trypanocidal Agents / Flavones / Medicinal Plant / DNA binding proteins / Lactones / Blood cells / Penaeidae / Blood Proteins / Molecular Structure / The American / Hemolysis / Lipopolysaccharide / Phytotherapy / Experimental parasitology / Humans / Infrared spectroscopy / Mice / Female / Animals / Natural Product / Male / Penaeus Monodon / Horseshoe crabs / Litopenaeus Vannamei / Peptides / Cyclic peptides / Selection Index / Antimicrobial Peptide / Chagas disease / Sesquiterpenes / T lymphocytes / Experimental / Infrared / Antimicrobial Cationic Peptides / Trypanosoma Cruzi / Cytotoxic Activity / Tritium / Eupatorium / Xenopus laevis / Antimicrobial agents / Mytilus edulis / Cutaneous Leishmaniasis / Veterinary Sciences / Trypanocidal Agents / Flavones / Medicinal Plant / DNA binding proteins / Lactones / Blood cells / Penaeidae / Blood Proteins / Molecular Structure / The American / Hemolysis
Pharmacological Characterization, Structural Studies, and In Vivo Activities of Anti-Chagas Disease Lead Compounds Derived from Tipifarnib
Microbiology / Medical Microbiology / Macromolecular X-Ray Crystallography / Humans / Mice / Female / Animals / Quinolones / Chagas disease / Trypanosoma Cruzi / Trypanocidal Agents / Triazoles / Structure activity Relationship / Female / Animals / Quinolones / Chagas disease / Trypanosoma Cruzi / Trypanocidal Agents / Triazoles / Structure activity Relationship
Trypanocidal Activity of Aziridinyl Nitrobenzamide Prodrugs
Microbiology / Medical Microbiology / Cercopithecus aethiops / Animals / Trypanosoma Cruzi / Trypanosoma brucei brucei / Antimicrobial agents / Trypanosomiasis / Trypanocidal Agents / Vero cells / Benzamides / Trypanosoma brucei brucei / Antimicrobial agents / Trypanosomiasis / Trypanocidal Agents / Vero cells / Benzamides
Antiparasitic activities of novel ruthenium/lapachol complexes
Inorganic Chemistry / Leishmania / Macromolecular X-Ray Crystallography / Humans / Mice / Animals / Naphthoquinones / Plasmodium falciparum / Antimalarials / Molecular Conformation / Trypanocidal Agents / Inorganic Biochemistry / Animals / Naphthoquinones / Plasmodium falciparum / Antimalarials / Molecular Conformation / Trypanocidal Agents / Inorganic Biochemistry
Antiparasitic activities of novel ruthenium/lapachol complexes
Inorganic Chemistry / Leishmania / Macromolecular X-Ray Crystallography / Humans / Mice / Animals / Naphthoquinones / Plasmodium falciparum / Antimalarials / Molecular Conformation / Trypanocidal Agents / Inorganic Biochemistry / Animals / Naphthoquinones / Plasmodium falciparum / Antimalarials / Molecular Conformation / Trypanocidal Agents / Inorganic Biochemistry
Vanadium polypyridyl compounds as potential antiparasitic and antitumoral agents: New achievements
Inorganic Chemistry / Leishmania / Inorganic / Apoptosis / DNA / Humans / Chagas disease / Vanadium / Trypanosoma Cruzi / Trypanocidal Agents / Inorganic Biochemistry / Structure activity Relationship / Cell Survival / Antineoplastic Agents / Humans / Chagas disease / Vanadium / Trypanosoma Cruzi / Trypanocidal Agents / Inorganic Biochemistry / Structure activity Relationship / Cell Survival / Antineoplastic Agents
Trypanosoma rangeli: Characterization of a Mg-dependent ecto ATP-diphosphohydrolase activity
Microbiology / Experimental parasitology / Animals / Lipoprotein(a) / Experimental / Trypanosoma / Veterinary Sciences / Trypanocidal Agents / Salivary Gland / Hydrolysis / Hydrogen-Ion Concentration / Sodium Fluoride / Adenosine Triphosphate / Trypanosoma / Veterinary Sciences / Trypanocidal Agents / Salivary Gland / Hydrolysis / Hydrogen-Ion Concentration / Sodium Fluoride / Adenosine Triphosphate
Trypanocidal Furamidine Analogues: Influence of Pyridine Nitrogens on Trypanocidal Activity, Transport Kinetics, and Resistance Patterns
Microbiology / Medical Microbiology / Female / Animals / Drug Resistance / Nitrogen / Rats / Pyridines / Antimicrobial agents / Trypanocidal Agents / Adenine / Pentamidine / Nitrogen / Rats / Pyridines / Antimicrobial agents / Trypanocidal Agents / Adenine / Pentamidine
Trypanocidal and Leishmanicidal Activities of Sesquiterpene Lactones from Ambrosia tenuifolia Sprengel (Asteraceae)
Microbiology / Medical Microbiology / Medicinal Plants / Phytotherapy / Experimental parasitology / Humans / Infrared spectroscopy / Mice / Female / Animals / Male / Horseshoe crabs / Peptides / Cyclic peptides / Selection Index / Chagas disease / Sesquiterpenes / Infrared / Antimicrobial Cationic Peptides / Trypanosoma Cruzi / Xenopus laevis / Antimicrobial agents / Mytilus edulis / Cutaneous Leishmaniasis / Veterinary Sciences / Trypanocidal Agents / DNA binding proteins / Lactones / Penaeidae / Blood Proteins / Molecular Structure / Hemolysis / Humans / Infrared spectroscopy / Mice / Female / Animals / Male / Horseshoe crabs / Peptides / Cyclic peptides / Selection Index / Chagas disease / Sesquiterpenes / Infrared / Antimicrobial Cationic Peptides / Trypanosoma Cruzi / Xenopus laevis / Antimicrobial agents / Mytilus edulis / Cutaneous Leishmaniasis / Veterinary Sciences / Trypanocidal Agents / DNA binding proteins / Lactones / Penaeidae / Blood Proteins / Molecular Structure / Hemolysis
Trypanosoma cruzi infection disturbs mitochondrial membrane potential and ROS production rate in cardiomyocytes
Mitochondria / Fluorescent Dyes and Reagents / Reactive Oxygen Species / Mice / Animals / Chagas disease / Enzyme / NADPH oxidase / IL / NOx / Rats / Trypanosoma Cruzi / Trypanocidal Agents / Inflammatory Cytokines / Mitochondrial Membrane Potential / Myeloperoxidase / Xanthine Oxidase / Biochemistry and cell biology / Production Rate / Chagas disease / Enzyme / NADPH oxidase / IL / NOx / Rats / Trypanosoma Cruzi / Trypanocidal Agents / Inflammatory Cytokines / Mitochondrial Membrane Potential / Myeloperoxidase / Xanthine Oxidase / Biochemistry and cell biology / Production Rate
In vitro antileishmanial, antiplasmodial and cytotoxic activities of phenolics and triterpenoids from Baccharis dracunculifolia D. C. (Asteraceae)
Complementary and Alternative Medicine / Plant Biology / Cytotoxicity / Propolis / Cercopithecus aethiops / Animals / Ursolic Acid / Phenols / Plant extracts / Cytotoxic Activity / Plasmodium falciparum / Antimalarials / Fitoterapia / Microbial Sensitivity Tests / Phytochemicals / Trypanocidal Agents / Vero cells / Triterpenoids / Baccharis / Triterpenes / Plant Leaves / Animals / Ursolic Acid / Phenols / Plant extracts / Cytotoxic Activity / Plasmodium falciparum / Antimalarials / Fitoterapia / Microbial Sensitivity Tests / Phytochemicals / Trypanocidal Agents / Vero cells / Triterpenoids / Baccharis / Triterpenes / Plant Leaves
Antitrypanosomal activities and cytotoxicity of 5-nitro-2-furancarbohydrazides
Organic Chemistry / Humans / Mice / Animals / Trypanosoma Cruzi / Trypanosoma brucei / Trypanosoma brucei brucei / Trypanocidal Agents / Leishmania infantum / Structure activity Relationship / Cell Survival / Trypanosoma brucei / Trypanosoma brucei brucei / Trypanocidal Agents / Leishmania infantum / Structure activity Relationship / Cell Survival
An in vitro iron superoxide dismutase inhibitor decreases the parasitemia levels of Trypanosoma cruzi in BALB/c mouse model during acute phase
Mice / Animals / Superoxide Dismutase / Chagas disease / Trypanosoma Cruzi / Immunocompromised host / Trypanocidal Agents / Cyclophosphamide / Molecular Structure / Immunocompromised host / Trypanocidal Agents / Cyclophosphamide / Molecular Structure
Cytotoxic, trypanocidal, and antifungal activities of Eugenia jambolana L
Nutrition and Dietetics / Macrophages / Mice / Animals / Candida / Antifungal Activity / Chagas disease / Plant extracts / Trypanosoma Cruzi / Antifungal Agents / Microbial Sensitivity Tests / Food Sciences / Medicinal Food / Trypanocidal Agents / Antiparasitic activity / Eugenia / Metronidazole / Cytotoxins / Plant Leaves / Antifungal Activity / Chagas disease / Plant extracts / Trypanosoma Cruzi / Antifungal Agents / Microbial Sensitivity Tests / Food Sciences / Medicinal Food / Trypanocidal Agents / Antiparasitic activity / Eugenia / Metronidazole / Cytotoxins / Plant Leaves
Trypanocide, cytotoxic, and antifungal activities of Momordica charantia
Traditional Medicine / Plant Biology / Macrophages / Cell line / Mice / Pharmaceutical / Animals / Candida / Antimicrobial activity / Antifungal Activity / Chagas disease / Pharmaceutical Biology / Plant extracts / Trypanosoma Cruzi / Antifungal Agents / Microbial Sensitivity Tests / Toxicity Tests / Momordica Charantia / Trypanocidal Agents / Antiparasitic activity / Metronidazole / Plant Leaves / Pharmaceutical / Animals / Candida / Antimicrobial activity / Antifungal Activity / Chagas disease / Pharmaceutical Biology / Plant extracts / Trypanosoma Cruzi / Antifungal Agents / Microbial Sensitivity Tests / Toxicity Tests / Momordica Charantia / Trypanocidal Agents / Antiparasitic activity / Metronidazole / Plant Leaves
Leishmanicidal Triterpenes from Lantana camara
Organic Chemistry / Humans / Lantana / Cutaneous Leishmaniasis / Trypanocidal Agents / Leishmania Major / Triterpenoids / Triterpenes / Plant Leaves / Leishmania Major / Triterpenoids / Triterpenes / Plant Leaves
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