Solubility

Danazol-β-cyclodextrin binary system: A potential application in emergency contraception by the oral route

Nuclear Magnetic Resonance / Magnetic Resonance Spectroscopy / Progesterone / Circular Dichroism / Mice / Female / Animals / Male / First-Order Logic / Solubility / Spectrum / Mouse Model / Emergency Contraception / AAPS PharmSciTech / Danazol / Female / Animals / Male / First-Order Logic / Solubility / Spectrum / Mouse Model / Emergency Contraception / AAPS PharmSciTech / Danazol

Iron Deficiency in Obese Postmenopausal Women*

Obesity / Multidisciplinary / Insulin Resistance / Postmenopausal Women / Humans / Regression Analysis / Transferrin / Research Method / Iron / Body Mass Index / Transferrin Receptor / Solubility / Multiple Regression / Children and Adolescents / Aged / Middle Aged / Iron status / Acute Phase Response / Control Group / Regression Analysis / Transferrin / Research Method / Iron / Body Mass Index / Transferrin Receptor / Solubility / Multiple Regression / Children and Adolescents / Aged / Middle Aged / Iron status / Acute Phase Response / Control Group

Iron Deficiency in Obese Postmenopausal Women

Obesity / Multidisciplinary / Insulin Resistance / Postmenopausal Women / Humans / Regression Analysis / Transferrin / Research Method / Iron / Body Mass Index / Transferrin Receptor / Solubility / Multiple Regression / Children and Adolescents / Aged / Middle Aged / Iron status / Acute Phase Response / Control Group / Regression Analysis / Transferrin / Research Method / Iron / Body Mass Index / Transferrin Receptor / Solubility / Multiple Regression / Children and Adolescents / Aged / Middle Aged / Iron status / Acute Phase Response / Control Group

Iron Deficiency in Obese Postmenopausal Women*

Obesity / Multidisciplinary / Insulin Resistance / Postmenopausal Women / Humans / Regression Analysis / Transferrin / Research Method / Iron / Body Mass Index / Transferrin Receptor / Solubility / Multiple Regression / Children and Adolescents / Aged / Middle Aged / Iron status / Acute Phase Response / Control Group / Regression Analysis / Transferrin / Research Method / Iron / Body Mass Index / Transferrin Receptor / Solubility / Multiple Regression / Children and Adolescents / Aged / Middle Aged / Iron status / Acute Phase Response / Control Group

Pro-apoptotic activity of α-bisabolol in preclinical models of primary human acute leukemia cells

Leukemia / Mitochondria / Adolescent / Apoptosis / Translational Medicine / Acute Myeloid Leukemia / Humans / Mutation / Female / Male / Cluster Analysis / Young Adult / Solubility / Sesquiterpenes / Lipid Raft / Middle Aged / Adult / Time Factors / Acute Lymphoid Leukemia / Culture Media / Mitochondrial Membrane Potential / Blood cells / Benzamides / Acute Myeloid Leukemia / Humans / Mutation / Female / Male / Cluster Analysis / Young Adult / Solubility / Sesquiterpenes / Lipid Raft / Middle Aged / Adult / Time Factors / Acute Lymphoid Leukemia / Culture Media / Mitochondrial Membrane Potential / Blood cells / Benzamides

Recombinant Plasmepsin 1 from the Human Malaria Parasite Plasmodium falciparum : Enzymatic Characterization, Active Site Inhibitor Design, and Structural Analysis

Biochemistry / Catalysis / Kinetics / Enzyme Inhibitors / Humans / Animals / Structure Analysis / Solubility / Active site / Substrate Specificity / Plasmodium falciparum / Protozoan Proteins / Amino Acid Sequence / Amino Acid Substitution Rates / Structure activity Relationship / Recombinant Proteins / Hydrogen-Ion Concentration / Biochemistry and cell biology / Molecular Structure / Molecular Sequence Data / Animals / Structure Analysis / Solubility / Active site / Substrate Specificity / Plasmodium falciparum / Protozoan Proteins / Amino Acid Sequence / Amino Acid Substitution Rates / Structure activity Relationship / Recombinant Proteins / Hydrogen-Ion Concentration / Biochemistry and cell biology / Molecular Structure / Molecular Sequence Data

Soy polysaccharide as a novel superdisintegrant in sildenafil citrate sublingual tablets: preparation, characterization, and in vivo evaluation

Pharmaceutical Technology / Polysaccharides / Pharmaceutical Chemistry / Humans / Wettability / Male / Hardness / Solubility / Phosphodiesterase Inhibitors / Soybeans / Adult / Tablets / Excipients / Drug Stability / Biological Availability / Male / Hardness / Solubility / Phosphodiesterase Inhibitors / Soybeans / Adult / Tablets / Excipients / Drug Stability / Biological Availability

A novel cholesterol transfer protein in cardiac sarcolemma. Purification and initial characterization

Western blotting / Cholesterol / Animals / Liposomes / Sodium Dodecyl Sulfate-Polyacrylamide Gel Electrophoresis / Solubility / Myocardium / Molecular weight / Rabbits / Plasma Membrane / Molecular and Cellular Biochemistry / Biochemistry and cell biology / Solubility / Myocardium / Molecular weight / Rabbits / Plasma Membrane / Molecular and Cellular Biochemistry / Biochemistry and cell biology

Biopharmaceutic evaluation of novel anthelmintic (1H-benzimidazol-5(6)-yl)carboxamide derivatives

Water / Pharmaceutics / Humans / Mice / Animals / Male / Solubility / Caco-2 cells / Anthelmintics / Benzimidazoles / Male / Solubility / Caco-2 cells / Anthelmintics / Benzimidazoles

Physicochemical and biopharmaceutical characterization ofendo-2-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-2,3-dihydro-1H-benz[e]isoindol-1-one (CR3124) a novel potent 5-HT3 receptor antagonist

Water / Scanning Electron Microscopy / Powder Diffraction / NMR Spectroscopy / Crystallization / Macromolecular X-Ray Crystallography / Molecular Dynamics / Crystal structure / Humans / Liver / Differential scanning calorimetry / Permeability / Pharmaceutical Sciences / Animals / Male / Solubility / Citrus / Intestinal absorption / Caco-2 cells / Rats / X ray diffraction / Carbon Tetrachloride / Molecular Conformation / Flavones / Drug Stability / Crystalline Structure / Drug Induced Liver Injury / Serotonin antagonists / Aspartate Aminotransferases / Alanine Transaminase / Macromolecular X-Ray Crystallography / Molecular Dynamics / Crystal structure / Humans / Liver / Differential scanning calorimetry / Permeability / Pharmaceutical Sciences / Animals / Male / Solubility / Citrus / Intestinal absorption / Caco-2 cells / Rats / X ray diffraction / Carbon Tetrachloride / Molecular Conformation / Flavones / Drug Stability / Crystalline Structure / Drug Induced Liver Injury / Serotonin antagonists / Aspartate Aminotransferases / Alanine Transaminase

Serum interleukin-6 receptor in polymyalgia rheumatica: A potential marker of relapse/recurrence risk

Psychology / Immunology / Multivariate Analysis / Clinical Practice / Humans / Female / Male / Risk factors / Solubility / Recurrence / Clinical Sciences / Aged / Middle Aged / Public health systems and services research / Prognosis / Biological markers / Risk Factors / Polymyalgia Rheumatica / Proportional Hazards Models / Female / Male / Risk factors / Solubility / Recurrence / Clinical Sciences / Aged / Middle Aged / Public health systems and services research / Prognosis / Biological markers / Risk Factors / Polymyalgia Rheumatica / Proportional Hazards Models

Precise protein solubility determination by Laser confocal differential interference contrast microscopy

Crystal Growth / Aqueous Solutions / Entropy / Enthalpy / Macromolecules / Proteins / Solubility / Macromolecule / Aqueous Solution / Differential Interference Contrast / Entropie / Proteins / Solubility / Macromolecule / Aqueous Solution / Differential Interference Contrast / Entropie

Physicochemical and biopharmaceutical characterization ofendo-2-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-2,3-dihydro-1H-benz[e]isoindol-1-one (CR3124) a novel potent 5-HT3 receptor antagonist

Water / Scanning Electron Microscopy / Powder Diffraction / NMR Spectroscopy / Crystallization / Macromolecular X-Ray Crystallography / Molecular Dynamics / Crystal structure / Humans / Liver / Differential scanning calorimetry / Permeability / Pharmaceutical Sciences / Animals / Male / Solubility / Citrus / Intestinal absorption / Caco-2 cells / Rats / X ray diffraction / Carbon Tetrachloride / Molecular Conformation / Flavones / Drug Stability / Crystalline Structure / Drug Induced Liver Injury / Serotonin antagonists / Aspartate Aminotransferases / Alanine Transaminase / Macromolecular X-Ray Crystallography / Molecular Dynamics / Crystal structure / Humans / Liver / Differential scanning calorimetry / Permeability / Pharmaceutical Sciences / Animals / Male / Solubility / Citrus / Intestinal absorption / Caco-2 cells / Rats / X ray diffraction / Carbon Tetrachloride / Molecular Conformation / Flavones / Drug Stability / Crystalline Structure / Drug Induced Liver Injury / Serotonin antagonists / Aspartate Aminotransferases / Alanine Transaminase

IL6/sIL6R complex contributes to emergency granulopoietic responses in G-CSF- and GM-CSF-deficient mice

Mice / Animals / Blood / Candida albicans / Solubility / Clinical Sciences / Neutrophils / Lipopolysaccharides / Monocytes / Survival Rate / Human Fibroblasts / Somatic Cell Count / Subcellular Fractions / Knockout Mice / Bone Marrow Cells / Interleukin / Clinical Sciences / Neutrophils / Lipopolysaccharides / Monocytes / Survival Rate / Human Fibroblasts / Somatic Cell Count / Subcellular Fractions / Knockout Mice / Bone Marrow Cells / Interleukin

Transition-State Analogue γ-Secretase Inhibitors Stabilize a 900 kDa Presenilin/Nicastrin Complex †

Biochemistry / Photochemistry / Membrane Proteins / Humans / Sodium Dodecyl Sulfate-Polyacrylamide Gel Electrophoresis / Solubility / Protease Inhibitors / Presenilin-2 / Molecular weight / Detergents / Subcellular Fractions / Protein Binding / Carbamates / Biochemistry and cell biology / Solubility / Protease Inhibitors / Presenilin-2 / Molecular weight / Detergents / Subcellular Fractions / Protein Binding / Carbamates / Biochemistry and cell biology

Novel composite core-shell nanoparticles as busulfan carriers

Biomedical Engineering / Complement activation / Pharmaceutical Technology / Drug delivery / Nanoparticles / Polymers / Pharmaceutical Chemistry / Controlled release / Solubility / Poly Ethylene Glycol / Surface Properties / Freeze Drying / Surface Charge / Chemical Composition / Liquid Scintillation Counting / Zeta Potential / Drug Carriers / Drug Release / Lactones / Cyanoacrylates / Polymers / Pharmaceutical Chemistry / Controlled release / Solubility / Poly Ethylene Glycol / Surface Properties / Freeze Drying / Surface Charge / Chemical Composition / Liquid Scintillation Counting / Zeta Potential / Drug Carriers / Drug Release / Lactones / Cyanoacrylates
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