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Organic Chemistry
Organic Chemistry
Benzylidene ketal derivatives as M2 muscarinic receptor antagonists
Organic Chemistry / Bioorganic and medicinal Chemistry / Muscarinic Receptor
Enhancement of pharmacokinetic properties and in vivo efficacy of benzylidene ketal M2 muscarinic receptor antagonists via benzamide modification
Organic Chemistry / Humans / Animals / Drug Design / Acetylcholine / Microdialysis / Rats / Bioorganic and medicinal Chemistry / Structure activity Relationship / Muscarinic Receptor / Area Under Curve / Benzamides / Microdialysis / Rats / Bioorganic and medicinal Chemistry / Structure activity Relationship / Muscarinic Receptor / Area Under Curve / Benzamides
2Aminomethyl piperidines as novel urotensin-II receptor antagonists
Organic Chemistry / Humans / G protein-coupled receptors / Bioorganic and medicinal Chemistry / Structure activity Relationship / Piperidines
Albizia procera gum as an excipient for oral controlled release matrix tablet
Organic Chemistry / Controlled release / Food Sciences / Carbohydrate Polymers
Secondary amines as new pharmacophores for macrofilaricidal drug design
Organic Chemistry / Amines / Female / Animals / Male / Drug Design / Filariasis / Muridae / Structure activity Relationship / Drug Design / Filariasis / Muridae / Structure activity Relationship
Parallel Synthesis and Anti-Malarial Activity of a Sulfonamide Library
Organic Chemistry / Fluorescence Microscopy / Cell line / Humans / Plasmodium falciparum / Antimalarials / Structure activity Relationship / Antimalarials / Structure activity Relationship
N-(4-Nitrophenylsulfonyl)- and N-(Fluorenylmethoxycarbonyl)-N-ethyl Amino Acid Methyl Esters - A Practical Approach
Organic Chemistry / Organic / Amino Acid Profile / Methyl Ester
Enantioselective esterase activity of an industrial glutaryl acylase
Organic Chemistry
Unusual antimalarial meroditerpenes from tropical red macroalgae
Organic Chemistry / Drug Discovery / Pharmacognosy / Structural Analysis / In Vitro / Humans / Circular Dichroism / Natural Product / Seaweed / Isolation / Absolute Configuration / Diterpenes / Plasmodium falciparum / Antimalarials / Conformational Analysis / Biological activity / Terpenoid / Humans / Circular Dichroism / Natural Product / Seaweed / Isolation / Absolute Configuration / Diterpenes / Plasmodium falciparum / Antimalarials / Conformational Analysis / Biological activity / Terpenoid
Sequence dependence of benzo[a]pyrene diol epoxide-DNA adduct conformer distribution: A study by laser-induced fluorescence/polyacrylamide gel electrophoresis
Inorganic Chemistry / Organic Chemistry / DNA / Lasers / Animals / Sodium Dodecyl Sulfate-Polyacrylamide Gel Electrophoresis / Laser Induced Fluorescence / Cattle / Base Sequence / Polyacrylamide Gel Electrophoresis / Food and Chemical Toxicology / Molecular Sequence Data / Sodium Dodecyl Sulfate-Polyacrylamide Gel Electrophoresis / Laser Induced Fluorescence / Cattle / Base Sequence / Polyacrylamide Gel Electrophoresis / Food and Chemical Toxicology / Molecular Sequence Data
ChemInform Abstract: Unusual Antimalarial Meroditerpenes from Tropical Red Macroalgae
Organic Chemistry / Drug Discovery / Pharmacognosy / Structural Analysis / In Vitro / Humans / Circular Dichroism / Natural Product / Seaweed / Isolation / Absolute Configuration / Diterpenes / Plasmodium falciparum / Antimalarials / Conformational Analysis / Biological activity / Terpenoid / Humans / Circular Dichroism / Natural Product / Seaweed / Isolation / Absolute Configuration / Diterpenes / Plasmodium falciparum / Antimalarials / Conformational Analysis / Biological activity / Terpenoid
Novel fungicidal benzylsulfanyl-phenylguanidines
Organic Chemistry / Caenorhabditis elegans / Biofilm / Animals / Sulfides / Bacteria / Candida albicans / Staphylococcus epidermidis / Antifungal Agents / Biological activity / Guanidines / Chemical Synthesis / Bactericidal Activity / Molecular Structure / Minimal Bactericidal Concentration / Bacteria / Candida albicans / Staphylococcus epidermidis / Antifungal Agents / Biological activity / Guanidines / Chemical Synthesis / Bactericidal Activity / Molecular Structure / Minimal Bactericidal Concentration
Unusual antimalarial meroditerpenes from tropical red macroalgae
Organic Chemistry / Drug Discovery / Pharmacognosy / Structural Analysis / In Vitro / Humans / Circular Dichroism / Natural Product / Seaweed / Isolation / Absolute Configuration / Diterpenes / Plasmodium falciparum / Antimalarials / Conformational Analysis / Biological activity / Terpenoid / Humans / Circular Dichroism / Natural Product / Seaweed / Isolation / Absolute Configuration / Diterpenes / Plasmodium falciparum / Antimalarials / Conformational Analysis / Biological activity / Terpenoid
Tumor-localizing and radiosensitizing properties of meso -tetra(4- nido -carboranylphenyl)porphyrin (H 2 TCP)
Organic Chemistry
Tumor-localizing and radiosensitizing properties of meso -tetra(4- nido -carboranylphenyl)porphyrin (H 2 TCP)
Organic Chemistry
In Vitro Leishmanicidal Activities of Sesquiterpene Lactones from Tithonia diversifolia against Leishmania braziliensis Promastigotes and Amastigotes
Organic Chemistry / Humans / Animals / Asteraceae / Sesquiterpenes / Molecules / Plant extracts / Cutaneous Leishmaniasis / Lactones / Plant Leaves / Molecules / Plant extracts / Cutaneous Leishmaniasis / Lactones / Plant Leaves
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