Organic Chemistry

Efficiency of off-axis astronomical adaptive systems: comparison of experimental data for different astronomical sites

Organic Chemistry / Adaptive Optics / Canary Islands / Adaptive System / Layered Structure / Experimental Data / Atmospheric Effects / Site testing / Experimental Data / Atmospheric Effects / Site testing

Efficiency of off-axis astronomical adaptive systems: comparison of experimental data for different astronomical sites

Organic Chemistry / Adaptive Optics / Canary Islands / Adaptive System / Layered Structure / Experimental Data / Atmospheric Effects / Site testing / Experimental Data / Atmospheric Effects / Site testing

In vitro and in vivo profile of 5-[(4′-trifluoromethyl-biphenyl-2-carbonyl)-amino]-1H-indole-2-carboxylic acid benzylmethyl carbamoylamide (dirlotapide), a novel potent MTP inhibitor for obesity

Organic Chemistry / Medicinal Chemistry / Obesity / Pharmacokinetics / Pharmaceutical Chemistry / Dogs / Cell line / In Vitro / Humans / Models / Animals / Drug Design / Enzyme / Food intake / In Vivo / Rats / Rat / Carboxylic Acids / Molecular Conformation / Bioorganic and medicinal Chemistry / Hydrogen-Ion Concentration / Chemical Synthesis / Carbamates / Selectivity / Dogs / Cell line / In Vitro / Humans / Models / Animals / Drug Design / Enzyme / Food intake / In Vivo / Rats / Rat / Carboxylic Acids / Molecular Conformation / Bioorganic and medicinal Chemistry / Hydrogen-Ion Concentration / Chemical Synthesis / Carbamates / Selectivity

Potential silicon-containing antifolates

Organic Chemistry / Transport Properties / Enzyme / Tetrahedron

In vivo active antimalarial isonitriles

Organic Chemistry / Porifera / Nitriles / Mice / Multidrug Resistance / Animals / Plasmodium falciparum / Antimalarials / Microbial Sensitivity Tests / Plasmodium yoelii / Structure activity Relationship / Animals / Plasmodium falciparum / Antimalarials / Microbial Sensitivity Tests / Plasmodium yoelii / Structure activity Relationship

Geraniol-derived 1,2,4-Trioxanes with potent in-vivo antimalarial activity

Organic Chemistry / Malaria / Mice / Animals / Terpenes / Antimalarials / Plasmodium yoelii / Multi Drug Resistant Cancer / Antimalarials / Plasmodium yoelii / Multi Drug Resistant Cancer

Geraniol-Derived 1,2,4-Trioxanes with Potent in vivo Antimalarial Activity

Organic Chemistry / Malaria / Mice / Animals / Terpenes / Antimalarials / Plasmodium yoelii / Multi Drug Resistant Cancer / Antimalarials / Plasmodium yoelii / Multi Drug Resistant Cancer

Structural characterization of cell wall polysaccharides from two plant species endemic to central Africa, Fleurya aestuans and Phragmenthera capitata

Organic Chemistry / Traditional Medicine / Time-of-flight mass spectrometry / Sequential Extraction / Gas Chromatography / Structure Analysis / Food Sciences / Plant species / Plant Cell Wall / Cell Wall / Carbohydrate / Carbohydrate Polymers / Structure Analysis / Food Sciences / Plant species / Plant Cell Wall / Cell Wall / Carbohydrate / Carbohydrate Polymers

Cinnamic Anilides as New Mitochondrial Permeability Transition Pore Inhibitors Endowed with Ischemia-Reperfusion Injury Protective Effect in Vivo

Organic Chemistry / Medicinal Chemistry / Calcium / Female / Animals / Male / Myocardial Infarction / Rabbits / Structure activity Relationship / Male / Myocardial Infarction / Rabbits / Structure activity Relationship

Enhancement of pharmacokinetic properties and in vivo efficacy of benzylidene ketal M2 muscarinic receptor antagonists via benzamide modification

Organic Chemistry / Pharmacokinetics / In Vitro / Humans / Animals / Drug Design / Acetylcholine / Bioavailability / Microdialysis / In Vivo / Rats / Rat / Cholinergic Receptor / Bioorganic and medicinal Chemistry / Structure activity Relationship / Muscarinic Receptor / Chemical Synthesis / Area Under Curve / Benzamides / Drug Design / Acetylcholine / Bioavailability / Microdialysis / In Vivo / Rats / Rat / Cholinergic Receptor / Bioorganic and medicinal Chemistry / Structure activity Relationship / Muscarinic Receptor / Chemical Synthesis / Area Under Curve / Benzamides
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