Nitriles

Extracellular signal-regulated kinase and GEF-H1 mediate depolarization-induced Rho activation and paracellular permeability increase

Physiology / Calcium / Enzyme Inhibitors / Flavonoids / Dogs / Nitriles / Permeability / Animals / Potassium / Phosphorylation / Medical Physiology / Organophosphorus Compounds / Epithelial cells / Time Factors / Swine / Transfection / Alanine / Protein Kinase Inhibitors / Biochemistry and cell biology / Ouabain / Nitriles / Permeability / Animals / Potassium / Phosphorylation / Medical Physiology / Organophosphorus Compounds / Epithelial cells / Time Factors / Swine / Transfection / Alanine / Protein Kinase Inhibitors / Biochemistry and cell biology / Ouabain

Effect of deltamethrin (pyrethroid insecticide) on two clones of Daphnia magna (Crustacea, Cladocera): A proteomic investigation

Aquatic Toxicology / Proteomics / Daphnia / Biological Sciences / Environmental Sciences / Nitriles / Animals / CHEMICAL SCIENCES / Biological markers / Gene Expression Regulation / Nitriles / Animals / CHEMICAL SCIENCES / Biological markers / Gene Expression Regulation

First Evidence of High Knockdown Resistance Frequency in Anopheles arabiensis (Diptera: Culicidae) from Ethiopia

Malaria / Tropical Medicine / Ethiopia / Insecticides / Insecticide Resistance / DDT / Nitriles / Anopheles / Resistance / Animals / Diptera / The American / Insect Vectors / DDT / Nitriles / Anopheles / Resistance / Animals / Diptera / The American / Insect Vectors

Acute effects of oestrogen receptor subtype-specific agonists on vascular contractility

British / Nitriles / Female / Animals / Male / Vasoconstriction / Phenols / Rats / Time Factors / Wistar Rats / Pyrazoles / Mesenteric Arteries / Estradiol / Estrogen receptor-beta / Selective estrogen receptor modulators / Estrogen receptor alpha / Vasoconstriction / Phenols / Rats / Time Factors / Wistar Rats / Pyrazoles / Mesenteric Arteries / Estradiol / Estrogen receptor-beta / Selective estrogen receptor modulators / Estrogen receptor alpha

Polycyclic dinitriles: a novel class of potent GABAergic insecticides provides a new radioligand, [3H]BIDN

Zoology / Invertebrate Neuroscience / Insecticides / Nitriles / GABA receptors / Animals / Molecular Modelling / Beetles / Radioligand Assay / Tritium / Invertebrate / Structure activity Relationship / Structural Similarity Index / Force Field Analysis / Pokemon / Neurosciences / GABA receptor / Animals / Molecular Modelling / Beetles / Radioligand Assay / Tritium / Invertebrate / Structure activity Relationship / Structural Similarity Index / Force Field Analysis / Pokemon / Neurosciences / GABA receptor

Systemic catechol-O-methyl transferase inhibition enables the D1 agonist radiotracer R-[11C]SKF 82957

Enzyme Inhibitors / Positron Emission Tomography / Brain / Nitriles / Animals / Benzophenones / Clinical Sciences / Rats / Catechols / Metabolic pathway / Radiopharmaceuticals / Benzophenones / Clinical Sciences / Rats / Catechols / Metabolic pathway / Radiopharmaceuticals

Insecticide resistance status in Anopheles culicifacies in Madhya Pradesh, central India

Survival Analysis / India / Insecticides / Insecticide Resistance / DDT / Nitriles / Anopheles / Female / Animals / VECTOR / Vector borne diseases / Malathion / Nitriles / Anopheles / Female / Animals / VECTOR / Vector borne diseases / Malathion

Polycyclic dinitriles: a novel class of potent GABAergic insecticides provides a new radioligand, [3H]BIDN

Zoology / Invertebrate Neuroscience / Insecticides / Nitriles / GABA receptors / Animals / Molecular Modelling / Beetles / Radioligand Assay / Tritium / Invertebrate / Structure activity Relationship / Structural Similarity Index / Force Field Analysis / Pokemon / Neurosciences / GABA receptor / Animals / Molecular Modelling / Beetles / Radioligand Assay / Tritium / Invertebrate / Structure activity Relationship / Structural Similarity Index / Force Field Analysis / Pokemon / Neurosciences / GABA receptor

Hypoxia sustains glioblastoma radioresistance through ERKs/DNA-PKcs/HIF-1α functional interplay

Oncology / Enzyme Inhibitors / Humans / Nitriles / Glioblastoma / Oxygen / Radiation Tolerance / Benzamides / Oxygen / Radiation Tolerance / Benzamides

Hydroxyflutamide enhances cellular sensitivity to 5-fluorouracil by suppressing thymidylate synthase expression in bicalutamide-resistant human prostate cancer cells

Oncology / Molecular Medicine / Cancer / Cell Cycle / Apoptosis / Humans / Nitriles / Cell / Male / Gene / Carcinoma / 5-FLUOROURACIL / Humans / Nitriles / Cell / Male / Gene / Carcinoma / 5-FLUOROURACIL

Datos de rilpivirina en pacientes naïve. Lecciones de los estudios ECHO, THRIVE y STaR

Medical Microbiology / Medication Adherence / Treatment Outcome / HIV / Safety / Humans / Nitriles / Female / Male / Efficacy / Adult / Combination drug therapy / Adverse effects / Viral Load / Multicenter Studies as Topic / Humans / Nitriles / Female / Male / Efficacy / Adult / Combination drug therapy / Adverse effects / Viral Load / Multicenter Studies as Topic

Entacapone, a novel catechol-O-methyltransferase inhibitor for Parkinson\'s disease, does not impair mitochondrial energy production

Kinetics / Enzyme Inhibitors / Mitochondria / Energy Metabolism / Cell Culture / Cell line / Nitriles / Mice / Female / Animals / Male / Heart / European / Energy Production / Rats / Oxidative phosphorylation / Guinea Pig / Catechols / Wistar Rats / Oxygen Consumption / Cardiac function / Cell line / Nitriles / Mice / Female / Animals / Male / Heart / European / Energy Production / Rats / Oxidative phosphorylation / Guinea Pig / Catechols / Wistar Rats / Oxygen Consumption / Cardiac function

Susceptibilidad de Aedes aegypti a DDT, deltametrina y lambdacialotrina en Colombia

Colorimetry / Colombia / Aedes aegypti / Insecticides / DDT / Nitriles / Animals / Drug Resistance / Acetylcholinesterase / Mosquito Control / Public health systems and services research / Biological Assay / Aedes / Nitriles / Animals / Drug Resistance / Acetylcholinesterase / Mosquito Control / Public health systems and services research / Biological Assay / Aedes

Susceptibilidad de Aedes aegypti a DDT, deltametrina y lambdacialotrina en Colombia

Colorimetry / Colombia / Aedes aegypti / Insecticides / DDT / Nitriles / Animals / Drug Resistance / Acetylcholinesterase / Mosquito Control / Public health systems and services research / Biological Assay / Aedes / Nitriles / Animals / Drug Resistance / Acetylcholinesterase / Mosquito Control / Public health systems and services research / Biological Assay / Aedes

Drug Approval Summaries: Arsenic Trioxide, Tamoxifen Citrate, Anastrazole, Paclitaxel, Bexarotene

Breast Cancer / Gene expression / Humans / Nitriles / Ductal carcinoma in situ / United States / Female / The / Paclitaxel / Arsenic trioxide / Tamoxifen / Triazoles / Oxides / Antineoplastic Agents / Arsenicals / Acute Promyelocytic Leukemia / Oncologist / cutaneous T-cell lymphoma / United States Food and Drug Administration / United States / Female / The / Paclitaxel / Arsenic trioxide / Tamoxifen / Triazoles / Oxides / Antineoplastic Agents / Arsenicals / Acute Promyelocytic Leukemia / Oncologist / cutaneous T-cell lymphoma / United States Food and Drug Administration
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