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Antimalarials
Antimalarials
Novel Conjugated Quinoline–Indoles Compromise Plasmodium falciparum Mitochondrial Function and Show Promising Antimalarial Activity
Organic Chemistry / Medicinal Chemistry / Mitochondria / Humans / Drug Resistance / Plasmodium falciparum / Antimalarials / Chloroquine / Structure activity Relationship / Hemoglobins / Plasmodium falciparum / Antimalarials / Chloroquine / Structure activity Relationship / Hemoglobins
Swedish traveller with Plasmodium knowlesi malaria after visiting Malaysian Borneo: a case report
Malaysia / Medical Microbiology / Malaria / Sweden / Travel / Humans / South east Asia / Animals / Male / Polymerase Chain Reaction / Differential Diagnosis / Borneo / Molecular Characterization / Adult / Antimalarials / Diagnostic Test / Sensitivity and Specificity / Plasmodium Knowlesi / Mefloquine / Humans / South east Asia / Animals / Male / Polymerase Chain Reaction / Differential Diagnosis / Borneo / Molecular Characterization / Adult / Antimalarials / Diagnostic Test / Sensitivity and Specificity / Plasmodium Knowlesi / Mefloquine
New Antimalarial Hits from Dacryodes edulis (Burseraceae) - Part I: Isolation, In Vitro Activity, In Silico “drug-likeness� and Pharmacokinetic Profiles
Drug interactions / Multidisciplinary / Cell line / Animals / PLoS one / Plant extracts / Epithelial cells / Plasmodium falciparum / Antimalarials / Toxicity Tests / Quinine / Plant extracts / Epithelial cells / Plasmodium falciparum / Antimalarials / Toxicity Tests / Quinine
Plasmodium falciparum neutral aminopeptidases: new targets for anti-malarials
Biological Sciences / Humans / CHEMICAL SCIENCES / Plasmodium falciparum / Antimalarials
Transient Lesion in the Splenium of the Corpus Callosum in Acute Uncomplicated Falciparum Malaria
Cognitive Science / Neurology / Eating Disorders / Magnetic Resonance Imaging / Epilepsy / Thailand / Electroencephalography / Adolescent / Prospective studies / Humans / Child / Corpus Callosum / Glioma / Female / Male / Young Adult / Follow-up studies / Thrombocytopenia / Clinical Sciences / Middle Aged / Adult / Carbamazepine / Antimalarials / Combination drug therapy / Medical Records / Chloroquine / X ray Computed Tomography / Neurosciences / Predictive value of tests / Brain Neoplasms / Primaquine / Hemolysis / Thailand / Electroencephalography / Adolescent / Prospective studies / Humans / Child / Corpus Callosum / Glioma / Female / Male / Young Adult / Follow-up studies / Thrombocytopenia / Clinical Sciences / Middle Aged / Adult / Carbamazepine / Antimalarials / Combination drug therapy / Medical Records / Chloroquine / X ray Computed Tomography / Neurosciences / Predictive value of tests / Brain Neoplasms / Primaquine / Hemolysis
Plasmodium vivax malaria relapses at a travel medicine centre in Rio de Janeiro, a non-endemic area in Brazil
Medical Microbiology / Malaria / Brazil / Adolescent / Humans / Female / Animals / Male / Young Adult / Risk factors / Recurrence / Middle Aged / Adult / Antimalarials / Risk Factors / Primaquine / Female / Animals / Male / Young Adult / Risk factors / Recurrence / Middle Aged / Adult / Antimalarials / Risk Factors / Primaquine
N -Aryl-2-aminobenzimidazoles: Novel, Efficacious, Antimalarial Lead Compounds
Pharmacology / Chemistry / Organic Chemistry / Pharmacy / Medicinal Chemistry / Malaria / Humans / Animals / Rats / Hepatocytes / Plasmodium falciparum / Antimalarials / Benzimidazoles / Structure activity Relationship / Plasmodium berghei / Malaria / Humans / Animals / Rats / Hepatocytes / Plasmodium falciparum / Antimalarials / Benzimidazoles / Structure activity Relationship / Plasmodium berghei
Antiplasmodial Alkaloids from Desmos rostrata
Natural Products / Medicinal Plants / Vietnam / Biological Sciences / Humans / Animals / Alkaloids / CHEMICAL SCIENCES / Plasmodium falciparum / Antimalarials / Natural / KB cells / Molecular Structure / Animals / Alkaloids / CHEMICAL SCIENCES / Plasmodium falciparum / Antimalarials / Natural / KB cells / Molecular Structure
Comparative insight into nucleotide excision repair components of Plasmodium falciparum
Genomics / DNA repair / Drug Resistance / Plasmodium falciparum / Antimalarials / Protozoan Proteins / Amino Acid Sequence / Biochemistry and cell biology / Protozoan Proteins / Amino Acid Sequence / Biochemistry and cell biology
The pharmacokinetic properties of intramuscular artesunate and rectal dihydroartemisinin in uncomplicated falciparum malaria
Nonparametric Statistics / British / Pharmacokinetics / Humans / Female / Male / Confidence intervals / Sesquiterpenes / Adult / Antimalarials / Cross-Over Studies / Area Under Curve / Male / Confidence intervals / Sesquiterpenes / Adult / Antimalarials / Cross-Over Studies / Area Under Curve
Fumagillin and Fumarranol Interact with P. falciparum Methionine Aminopeptidase 2 and Inhibit Malaria Parasite Growth In Vitro and In Vivo
Organic Chemistry / Malaria / Saccharomyces cerevisiae / Humans / Sequence alignment / Escherichia coli / Mice / Female / Animals / Sesquiterpenes / Plasmodium falciparum / Antimalarials / Protozoan Proteins / Cell Proliferation / Amino Acid Sequence / Chemistry Biology / Recombinant Proteins / Protein Binding / Biochemistry and cell biology / Escherichia coli / Mice / Female / Animals / Sesquiterpenes / Plasmodium falciparum / Antimalarials / Protozoan Proteins / Cell Proliferation / Amino Acid Sequence / Chemistry Biology / Recombinant Proteins / Protein Binding / Biochemistry and cell biology
Mefloquine pharmacokinetics and mefloquine-artesunate effectiveness in Peruvian patients with uncomplicated Plasmodium falciparum malaria
Medical Microbiology / Malaria / Peru / Treatment Outcome / Adolescent / Humans / Female / Animals / Blood sampling / Male / Young Adult / High Performance Liquid Chromatography / High Pressure Liquid Chromatography / Middle Aged / Adult / Ethnic Group / Time Factors / Plasmodium falciparum / Antimalarials / Combination drug therapy / Mefloquine / Humans / Female / Animals / Blood sampling / Male / Young Adult / High Performance Liquid Chromatography / High Pressure Liquid Chromatography / Middle Aged / Adult / Ethnic Group / Time Factors / Plasmodium falciparum / Antimalarials / Combination drug therapy / Mefloquine
Spatial distribution of G6PD deficiency variants across malaria-endemic regions
Spatial Analysis / Global Health / Medical Microbiology / Malaria / Risk assessment / Humans / Antimalarials / Genetic variation / Risk Assessment / Primaquine / Humans / Antimalarials / Genetic variation / Risk Assessment / Primaquine
Spatial distribution of G6PD deficiency variants across malaria-endemic regions
Spatial Analysis / Global Health / Medical Microbiology / Malaria / Risk assessment / Humans / Antimalarials / Genetic variation / Risk Assessment / Primaquine / Humans / Antimalarials / Genetic variation / Risk Assessment / Primaquine
Efficacy of Proveblue (Methylene Blue) in an Experimental Cerebral Malaria Murine Model
Microbiology / Medical Microbiology / Enzyme Inhibitors / Mice / Female / Animals / Methylene Blue / Antimalarials / Combination drug therapy / Cerebral Malaria / Plasmodium berghei / Animals / Methylene Blue / Antimalarials / Combination drug therapy / Cerebral Malaria / Plasmodium berghei
Amino derivatives of indolone-N-oxide: Preparation and antiplasmodial properties
Organic Chemistry / Mass Spectrometry / Magnetic Resonance Spectroscopy / Animals / Plasmodium falciparum / Antimalarials / Oxides / Antimalarials / Oxides
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